On-chip fragment-based approach for discovery of high-affinity bivalent inhibitors

Chembiochem. 2009 Mar 23;10(5):838-43. doi: 10.1002/cbic.200800704.
No abstract available

Publication types

  • Evaluation Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Cell Line
  • Drug Discovery
  • Humans
  • Immunosuppressive Agents / chemistry
  • Immunosuppressive Agents / metabolism
  • Ligands*
  • Molecular Structure
  • Peptide Fragments / chemistry
  • Peptide Fragments / metabolism*
  • Protein Array Analysis* / instrumentation
  • Protein Array Analysis* / methods
  • Protein Binding
  • Proteins / chemistry
  • Proteins / metabolism*
  • Tacrolimus / chemistry
  • Tacrolimus / metabolism
  • Tacrolimus Binding Protein 1A / genetics
  • Tacrolimus Binding Protein 1A / metabolism

Substances

  • Immunosuppressive Agents
  • Ligands
  • Peptide Fragments
  • Proteins
  • Tacrolimus Binding Protein 1A
  • Tacrolimus